Butidrine

Chemical compound From Wikipedia, the free encyclopedia

Butidrine (INNTooltip International Nonproprietary Name), sold under the brand names Betabloc, Butidrate, and Recetan among others, is a beta blocker (or β-adrenergic receptor antagonist) related to pronethalol[1] and propranolol[2] that was developed in the 1960s.[3][4] It is not cardioselective (i.e., is not selective for the β1-adrenergic receptor over the β2-adrenergic receptor).[5] It has membrane stabilizing activity but no intrinsic sympathomimetic activity (i.e., partial agonist activity).[6] Similarly to certain other beta blockers, butidrine additionally possesses local anesthetic properties.[7]

Trade namesBetabloc, Butidrate, Recetan
Other namesButedrine; Butydrine; Hydrobutamine; Idrobutamine
CAS Number
Quick facts Clinical data, Trade names ...
Butidrine
Clinical data
Trade namesBetabloc, Butidrate, Recetan
Other namesButedrine; Butydrine; Hydrobutamine; Idrobutamine
Drug classBeta blocker
Identifiers
  • 2-(butan-2-ylamino)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethanol
CAS Number
PubChem CID
ChemSpider
UNII
ChEBI
ChEMBL
CompTox Dashboard (EPA)
Chemical and physical data
FormulaC16H25NO
Molar mass247.382 g·mol−1
3D model (JSmol)
  • CCC(C)NCC(C1=CC2=C(CCCC2)C=C1)O
  • InChI=1S/C16H25NO/c1-3-12(2)17-11-16(18)15-9-8-13-6-4-5-7-14(13)10-15/h8-10,12,16-18H,3-7,11H2,1-2H3
  • Key:GVNYSERWAKVROD-UHFFFAOYSA-N
Close

References

Related Articles

Wikiwand AI