DLX-2270

Chemical compound From Wikipedia, the free encyclopedia

DLX-2270 is an experimental serotonin receptor modulator which is under investigation for the potential treatment of schizophrenia.[1]

Other namesDLX2270
ATC code
  • None
Quick facts Clinical data, Other names ...
DLX-2270
Clinical data
Other namesDLX2270
Routes of
administration
Oral[1]
Drug classSerotonin 5-HT2A receptor antagonist; Serotonin 5-HT2C receptor agonist; Antipsychotic; Psychoplastogen[1]
ATC code
  • None
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It acts as a serotonin 5-HT2A receptor antagonist and serotonin 5-HT2C receptor agonist.[1] In contrast to conventional antipsychotics, DLX-2270 is not a dopamine D2 receptor antagonist.[1] The drug is orally active and centrally penetrant.[1] In preclinical research, DLX-2270 has psychoplastogenic effects.[1] It reverses hyperlocomotion and social interaction deficits induced by the NMDA receptor antagonist phencyclidine (PCP).[1] In contrast to serotonin 5-HT2A receptor agonists, DLX-2270 does not produce the head-twitch response in rodents, and hence would not be expected to be hallucinogenic in humans.[1]

DLX-2270 was first described in the scientific literature in 2025.[1] It is under development by Delix Therapeutics.[1] DLX-2270 is a small molecule, but its chemical structure does not yet appear to have been disclosed.[1]

See also

References

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