Anazocine

Anazocine (INN; also known as azabicyclane or CS-307) is an opioid analgesic of the morphan/benzomorphan family developed in the middle 1960s in the United States which was never marketed.^[1][2]

ATC code

• None

CAS Number

• 15378-99-1
  21650-02-2 (citrate)

PubChem CID

• 27213

ChemSpider

• 25327

Quick facts Clinical data, ATC code ...

Anazocine

Clinical data
ATC code	None
Identifiers
IUPAC name 9-Methoxy-3-methyl-9-phenyl-3-azabicyclo[3.3.1]nonane
CAS Number	15378-99-1 21650-02-2 (citrate)
PubChem CID	27213
ChemSpider	25327
UNII	K2S5VMM2SG
ChEMBL	ChEMBL2105792
CompTox Dashboard (EPA)	DTXSID30864591
Chemical and physical data
Formula	C16H23NO
Molar mass	245.366 g·mol−1
3D model (JSmol)	Interactive image
SMILES O(C2(c1ccccc1)C3CCCC2CN(C3)C)C
InChI InChI=1S/C16H23NO/c1-17-11-14-9-6-10-15(12-17)16(14,18-2)13-7-4-3-5-8-13/h3-5,7-8,14-15H,6,9-12H2,1-2H3 Key:YFFNPIAPUDUYAU-UHFFFAOYSA-N

Close

The structure and properties of several related α- and β-azabicyclane opioids was explored.^[3] Anazocine's chemical and structural relatives include opioid partial agonists, mixed agonist-antagonists, pure agonists, antagonists, and atypical non-opioid analgesics. It was tested in pigeons and in other experiments which contrasted and compared its analgesic effects to those of the phenazepine opioid ethoheptazine and the phenalkoxam open chain opioid propoxyphene,^[4] and pethidine as well.^[5]