SER-601

SER-601 (COR-167) is a drug which acts as a potent and selective cannabinoid CB₂ receptor agonist, based on a quinolone-3-carboxylic acid core structure, with 190 times selectivity for CB₂ over the related CB₁ receptor. It has analgesic effects in animal studies, as well as neuroprotective effects,^[1] but without a "cannabis high" due to its low affinity for CB₁.^[2] A number of related compounds are known, almost all of which have high selectivity for CB₂.^[3]

Routes of
administrationOral

CAS Number

• 1048038-90-9 ^Y

PubChem CID

• 25034551

ChemSpider

• 24606023 ^Y

Quick facts Clinical data, Routes ofadministration ...

SER-601

Clinical data
Routes of administration	Oral
Identifiers
IUPAC name N-(Adamant-1-yl)-1-pentyl-4-oxo-6-isopropyl-1,4-dihydroquinoline-3-carboxamide
CAS Number	1048038-90-9 Y
PubChem CID	25034551
ChemSpider	24606023 Y
UNII	S723GJY405
ChEMBL	ChEMBL502276 Y
CompTox Dashboard (EPA)	DTXSID80648525
Chemical and physical data
Formula	C28H38N2O2
Molar mass	434.624 g·mol−1
3D model (JSmol)	Interactive image
SMILES CC(C)c5ccc(c1c5)n(CCCCC)cc(c1=O)C(=O)NC4(C2)CC(CC2C3)CC3C4
InChI InChI=1S/C28H38N2O2/c1-4-5-6-9-30-17-24(26(31)23-13-22(18(2)3)7-8-25(23)30)27(32)29-28-14-19-10-20(15-28)12-21(11-19)16-28/h7-8,13,17-21H,4-6,9-12,14-16H2,1-3H3,(H,29,32) Y Key:KUMKLUDNETVLDS-UHFFFAOYSA-N Y
NY (what is this?)  (verify)

Close