Tertatolol

Tertatolol (Artex, Artexal, Prenalex) is a medication in the class of beta blockers, used in the treatment of high blood pressure. It was discovered by the French pharmaceutical company Servier and is marketed in Europe.^[1]

AHFS/Drugs.comInternational Drug Names

Routes of
administrationOral

ATC code

• C07AA16 (WHO)

Legal status

• In general: ℞ (Prescription only)

Quick facts Clinical data, AHFS/Drugs.com ...

Tertatolol

Clinical data
AHFS/Drugs.com	International Drug Names
Routes of administration	Oral
ATC code	C07AA16 (WHO)
Legal status
Legal status	In general: ℞ (Prescription only)
Identifiers
IUPAC name (±)-1-(tert-Butylamino)-3-(3,4-dihydro-2H-thiochromen-8-yloxy)propan-2-ol
CAS Number	83688-84-0 Y
PubChem CID	36920
IUPHAR/BPS	571
ChemSpider	33875 N
UNII	9ZO341YQXP
KEGG	D07182 Y
ChEMBL	ChEMBL434200 N
CompTox Dashboard (EPA)	DTXSID80865735
ECHA InfoCard	100.073.179
Chemical and physical data
Formula	C16H25NO2S
Molar mass	295.44 g·mol−1
3D model (JSmol)	Interactive image
Chirality	Racemic mixture
SMILES CC(C)(C)NCC(COC1=CC=CC2=C1SCCC2)O
InChI InChI=1S/C16H25NO2S/c1-16(2,3)17-10-13(18)11-19-14-8-4-6-12-7-5-9-20-15(12)14/h4,6,8,13,17-18H,5,7,9-11H2,1-3H3 N Key:HTWFXPCUFWKXOP-UHFFFAOYSA-N N
NY (what is this?)  (verify)

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Tertatolol produces unique renal vasodilatory effects, mostly at a microcirculatory level, and inhibits human mesangial cell proliferation.^[2] Tertatolol has also been shown to act as a serotonin 5-HT_1A and 5-HT_1B receptor antagonist, similarly to propranolol and pindolol.^[3][4][5]