ADCYAP1R1

Protein-coding gene in the species Homo sapiens From Wikipedia, the free encyclopedia

Pituitary adenylate cyclase-activating polypeptide type I receptor also known as PAC1, is a protein that in humans is encoded by the ADCYAP1R1 gene.[5] This receptor binds pituitary adenylate cyclase activating peptide.[6][7]

PDBOrtholog search: PDBe RCSB
AliasesADCYAP1R1, PAC1, PAC1R, PACAPR, PACAPRI, ADCYAP receptor type I
Quick facts Available structures, PDB ...
ADCYAP1R1
Available structures
PDBOrtholog search: PDBe RCSB
Identifiers
AliasesADCYAP1R1, PAC1, PAC1R, PACAPR, PACAPRI, ADCYAP receptor type I
External IDsOMIM: 102981; MGI: 108449; HomoloGene: 870; GeneCards: ADCYAP1R1; OMA:ADCYAP1R1 - orthologs
Orthologs
SpeciesHumanMouse
Entrez
Ensembl
UniProt
RefSeq (mRNA)

NM_001118
NM_001199635
NM_001199636
NM_001199637

NM_001025372
NM_007407

RefSeq (protein)

NP_001109
NP_001186564
NP_001186565
NP_001186566

NP_001020543
NP_031433

Location (UCSC)Chr 7: 31.05 – 31.11 MbChr 6: 55.43 – 55.48 Mb
PubMed search[3][4]
Wikidata
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Function

PAC1 is a membrane-associated protein and shares significant homology with members of the G-protein coupled class B glucagon/secretin receptor family.[8] This receptor mediates diverse biological actions of adenylate cyclase activating polypeptide 1 and is positively coupled to adenylate cyclase. Alternative splicing of two exons of this gene generates four major splice variants, but their full-length nature has not been determined.[5] PAC1 is expressed in the adrenal medulla, pancreatic acini, uterus, myenteric plexus and brain.[9][10][11] It is also expressed in the trigeminal, otic and superior cervical ganglia (prejunctional) and cerebral arteries (postjunctional).[12]

Ligands

Agonists
  • PACAP-38 (endogenous peptide agonist, full length version) - also activates other receptors VIP, GPR55 and MRGPRX2 and the Secretin receptor.[13]
  • PACAP-27 (endogenous peptide agonist, shorter fragment which retains activity)
Antagonists

References

Further reading

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